What is Granisetron: Uses, Warnings & Interactions

Updated May 14, 2025  •  Published Dec 30, 2020

Granisetron overview

BRAND NAMES:

  • Kytril, Granisol

Generic Names:

  • Granisetron Hcl

Uses:

  • Treats nausea and vomiting caused by cancer treatments (chemotherapy or radiation).

Therapeutic Classes:

  • Antiemetic

Forms:

  • Tablet, Solution

How it’s taken:

  • By mouth

What is Granisetron used for?

What form(s) does Granisetron come in

  • Tablet

  • Solution

What are common Granisetron doses?

  • Tablet 1MG

  • Vial 1ML of 1MG/ML

  • Box 2 Tablets

Common Granisetron prescriptions

  • Granisetron HCl
    2 tablets box

  • Granisetron HCl
    1mg tablet

  • Granisetron HCl
    1ml of 1mg/ml vial

  • Granisetron HCl
    4ml of 4mg/4ml vial

How to take Granisetron

  • Your doctor will tell you how much medicine to use. Do not use more than directed. You will take this medicine only on the days you have your cancer treatment.

  • Measure the oral liquid medicine with a marked measuring spoon, oral syringe, or medicine cup.

  • Oral routeIt is best to take this medicine with food or milk.

  • Measure the oral liquid medicine with a marked measuring spoon, oral syringe, or medicine cup.

  • Your doctor will tell you how much medicine to use. Do not use more than directed. You will take this medicine only on the days you have your cancer treatment.

  • Oral routeIt is best to take this medicine with food or milk.

What to do if you miss a dose of Granisetron

  • Take a dose as soon as you remember. If it is almost time for your next dose, wait until then and take a regular dose. Do not take extra medicine to make up for a missed dose.

  • Keep all medicine out of the reach of children. Never share your medicine with anyone.

  • Ask your pharmacist, doctor, or health caregiver about the best way to dispose of any outdated medicine or medicine no longer needed.

Granisetron contraindications

  • You should not use this medicine if you have had an allergic reaction to granisetron.

Granisetron warnings

  • Make sure your doctor knows if you are pregnant or breast feeding.

Granisetron interactions

  • Make sure your doctor knows if you are pregnant or breast feeding.

Granisetron side effects

Serious Side Effects

  • Allergic reaction: Itching or hives, swelling in your face or hands, swelling or tingling in your mouth or throat, chest tightness, trouble breathing

  • Feeling unusually tired, weak, or anxious.

  • Fever.

  • Headache.

  • Lightheadedness, dizziness, or fainting.

  • Stomach pain, upset stomach, constipation, or diarrhea.

  • Unable to sleep, or feeling overly sleepy.

Less Serious Side Effects

  • Fever.

  • Chest pain.

  • Unable to sleep, or feeling overly sleepy.

  • Headache.

  • Feeling unusually tired, weak, or anxious.

  • Lightheadedness, dizziness, or fainting.

  • Stomach pain, upset stomach, constipation, or diarrhea.

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