Akynzeo is a prescription drug used in combination with dexamethasone to relieve nausea or delayed nausea due to cancer chemotherapy. Helsinn Therapeutics makes this medication. Akynzeo is available in two formulations: an oral capsule and an injection. Akynzeo works by blocking substances in the body and brain that cause nausea and vomiting. The retail price for Akynzeo is $849.82 for 1, 235-0.25mg solution reconstituted, a coupon from the SingleCare Akynzeo discount program reduces the price of Akynzeo to $670.15 for 1, 235-0.25mg solution reconstituted at major pharmacies nationwide.
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Los precios de los medicamentos recetados de SingleCare se basan en diversas fuentes. Los precios que publicamos son nuestra mejor estimación, pero no podemos garantizar que el precio que mostramos coincida exactamente con el precio que recibes en la farmacia. Para saber el precio exacto, por favor, comunícate con tu farmacia y proporciona los números BIN/GRP/PCN que aparecen en tu tarjeta de SingleCare.
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Precios actualizados: 05/12/2025
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Akynzeo is a prescription drug used in combination with dexamethasone to relieve nausea or delayed nausea due to cancer chemotherapy. Helsinn Therapeutics makes this medication. Akynzeo is available in two formulations: an oral capsule and an injection. Akynzeo works by blocking substances in the body and brain that cause nausea and vomiting. The retail price for Akynzeo is $849.82 for 1, 235-0.25mg solution reconstituted, a coupon from the SingleCare Akynzeo discount program reduces the price of Akynzeo to $670.15 for 1, 235-0.25mg solution reconstituted at major pharmacies nationwide.
Akynzeo is a prescription drug used in combination with dexamethasone to relieve nausea or delayed nausea due to cancer chemotherapy. Helsinn Therapeutics makes this medication. Akynzeo is available in two formulations: an oral capsule and an injection. Akynzeo works by blocking substances in the body and brain that cause nausea and vomiting. The retail price for Akynzeo is $849.82 for 1, 235-0.25mg solution reconstituted, a coupon from the SingleCare Akynzeo discount program reduces the price of Akynzeo to $670.15 for 1, 235-0.25mg solution reconstituted at major pharmacies nationwide.
Consumers will pay an average of $849.82 for 1, 235-0.25mg solution reconstituted of Akynzeo without insurance, but the price may vary by pharmacy. The cost for Akynzeo is $670.15 for 1, 235-0.25mg solution reconstituted with a SingleCare Akynzeo coupon. There are no eligibility criteria required to use a SingleCare discount for prescription savings. All you need to do is present a valid prescription at a local participating pharmacy in the United States. Check the SingleCare website to start saving.
Akynzeo copay costs may vary depending on specific insurance carriers. With SingleCare, Akynzeo costs $670.15 for 1, 235-0.25mg solution reconstituted. You can ask your pharmacist to compare the SingleCare price with your cost using insurance. A SingleCare savings card typically saves individuals up to 80% off on prescription drugs, which may be lower than the copay.
Akynzeo is usually not covered by Medicare prescription drug plans but may be covered by Medicare Part B, especially if the medication is given at a healthcare facility.
Akynzeo is a brand-name prescription drug in an oral capsule (netupitant and palonosetron) or intravenous form (fosnetupitant and palonosetron). No generic versions of Akynzeo are currently available.
Akynzeo is a medication prescribed to adults (in combination with a steroid medicine called dexamethasone) to relieve nausea due to cancer chemotherapy. Akynzeo is available in two formulations. The oral capsule form contains the active ingredients netupitant and palonosetron. The injection form contains the active ingredients fosnetupitant and palonosetron. Netupitant and fosnetupitant are classified as substance P/neurokinin-1 receptor antagonists, and palonosetron is a serotonin receptor antagonist.
Akynzeo works by blocking substances in the body and brain that cause nausea and vomiting.
Akynzeo is administered as a capsule (netupitant and palonosetron) or intravenous injection (fosnetupitant and palonosetron). The capsule is administered one hour before chemotherapy and the intravenous injection 30 minutes before chemotherapy.
Common adverse effects of Akynzeo include but are not limited to, headache, weakness, fatigue, constipation, and indigestion.
Allergic reactions are not common but can be severe and life-threatening. Patients who have symptoms of an allergic reaction, including hives, swelling, or trouble breathing, should get emergency medical attention.
This is not a complete list of possible side effects. You should consult with your prescribing physician about possible side effects of Akynzeo and any other concerns you may have.
Before taking Akynzeo, tell your healthcare provider about all the medications you take, including prescription and OTC drugs, vitamins, and supplements. While taking this medicine, do not take any new medications unless approved by your doctor. Some examples of drug interactions include:
Xanax (alprazolam)
Certain chemotherapy drugs
Rifampin
Nizoral (ketoconazole)
Concomitant use of medicines that increase serotonin levels—including SSRI antidepressants such as Lexapro (escitalopram) or SNRI antidepressants such as Cymbalta (duloxetine)—cause an increased risk of serotonin syndrome, a life-threatening condition caused by the buildup of excess serotonin
This is not a full list of drug interactions. Consult your healthcare professional for more information, questions, and medical advice on drug interactions.
Akynzeo in oral capsule form is taken as one capsule by mouth one hour before chemotherapy, along with a corticosteroid medicine called dexamethasone.
If given by intravenous infusion, Akynzeo is given as a one-time dose starting 30 minutes before chemotherapy and infused over 30 minutes. It is also given along with dexamethasone.
Consult your healthcare provider for more information or questions about taking this medicine.
After receiving her doctorate from the University of Pittsburgh School of Pharmacy, Karen Berger, Pharm.D., has worked in both chain and independent community pharmacies. She currently works at an independent pharmacy in New Jersey. Dr. Berger enjoys helping patients understand medical conditions and medications—both in person as a pharmacist, and online as a medical writer and reviewer.
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